pan-BET/BD2-IN-1
pan-BET/BD2-IN-1 (compound 6b) is a selective extra-terminal (BET) protein inhibitor (BRDT-1 Ki = 1.05 μM and BRD4-1 Ki = 0.68 μM). pan-BET/BD2-IN-1 inhibits MM.1S cancer cell growth with an IC50 of 2.6 μM.
For research use only. We do not sell to patients.
- Formula: C27H27N3O6
- Molecular Weight:489.52
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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Molecular Weight 489.52
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Formula C27H27N3O6
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SMILES
CC1=CC=C(C(OCCOC2=C(C=CC=C2)COC3=O)=C1)C4C3=C(NC(N(C(N5)=O)CC)=C4C5=O)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)