219 Results for "

Decyclohexanamine-Exatecan

" in MedChemExpress (MCE) Product Catalog:
Products (219)

219 Results for "Decyclohexanamine-Exatecan" in MCE Product Catalog:

Cat. No.: HY-P5287
CAS No.: 393781-65-2
Target:  

Integrin

Research Areas:  

Cancer

cRGDfK-thioacetyl ester is a bioactive polypeptide molecule. cRGDfK peptide has a selective affinity for integrins. cRGDfK peptide can modify NIR fluorescent probes for cancer targeting imaging .
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Cat. No.: HY-P5287A
Target:  

Integrin

Research Areas:  

Cancer

cRGDfK-thioacetyl ester TFA is a bioactive polypeptide molecule. cRGDfK peptide has a selective affinity for integrins. cRGDfK peptide can modify NIR fluorescent probes for cancer targeting imaging .
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Cat. No.: HY-P5643
CAS No.: 724760-20-7
Target:  

Bacterial

Research Areas:  

Infection

Retrocyclin-2 is an antimicrobial peptide against human immunodeficiency virus, influenza A and herpes simplex virus .
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Cat. No.: HY-P5644
CAS No.: 724760-21-8
Target:  

Bacterial

Research Areas:  

Infection

Retrocyclin-3 is an antimicrobial peptide against human immunodeficiency virus, influenza A and herpes simplex virus .
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Cat. No.: HY-P5997
CAS No.: 2104728-28-9
XQ2B is a specific cGAS inhibitor targeting protein-DNA interaction and phase separation. XQ2B markedly reduces ISD-induced Autophagy. XQ2B inhibits herpes simplex virus 1 (HSV-1)-induced antiviral immune responses and enhances HSV-1 infection .
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Cat. No.: HY-W019721
CAS No.: 63775-96-2
Cyclosporin D, a metabolite of Cyclosporin A, is a weak immunosuppressant. Cyclosporin D is used as internal standard for quantification of Cyclosporin A . Cyclosporin A is a potent immunosuppressant agent, suppress T cell activation by inhibiting calcineurin and the calcineurin-dependent transcription factors nuclear factor of activated T cells (NFAc) .
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Cat. No.: HY-106103
CAS No.: 81377-02-8
Purity:  99.30%
Synonyms: MK-678; L-363586
Seglitide (MK-678) is an orally active, selective SSTR2 agonist and somatostatin analog. Seglitide also acts as a competitive Somatostatin receptor antagonist, with pA2 values of 6.50, 6.24 and 6.09 against SS14, SS25 and SS28, respectively. Seglitide produces only weak, transient inhibition of myocardial contractility in isolated right atria of guinea pigs. Seglitide inhibits glucagon secretion and reduces circulating insulin levels. Seglitide causes a sustained, reversible reduction in elevated systolic blood pressure in streptozotocin (HY-13753)-induced diabetic rats, but exerts no effect on spontaneously hypertensive rats. Seglitide induces membrane hyperpolarization and inhibits electrical excitability. Seglitide induces concentration-dependent contraction and significant desensitization in isolated distal colon of rats. Seglitide can be used in research related to hypertension complicated with insulin-dependent diabetes mellitus .
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Cat. No.: HY-106103A
CAS No.: 99248-33-6
Purity:  99.30%
Synonyms: MK 678 acetate; L 36358 acetate
Seglitide acetate (MK 678; L 36358 acetate) is a potent, orally active somatostatin receptor 2 (SSTR2) agonist, and also a competitive antagonist of SSTR14, SSTR25, and SSTR28. Seglitide acetate has antihypertensive effects and can inhibit plasma glucagon and growth hormone. Seglitide acetate can be used for research on diabetes .
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Cat. No.: HY-146127
CAS No.: 3069455-54-2
Target:  

MEK

Research Areas:  

Cancer

Grb2 SH2 domain inhibitor 1 is an inhibitor of the Grb2 SH2 domain with an IC50 of 0.40 μM. Grb2 SH2 domain inhibitor 1 is also a cell-permeable cyclic peptide that can enter the cytosol of mammalian cells. Grb2 SH2 domain inhibitor 1 downregulates the expression level of p-MEK. Grb2 SH2 domain inhibitor 1 can be used in the research of breast cancer .
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Cat. No.: HY-146127A
Purity:  99.71%
Target:  

Src

Research Areas:  

Others

Grb2 SH2 domain inhibitor 1 TFA is a conformationally restricted cyclic cell penetrating peptide (CPP) containing d-pro-l-pro motif ring (AF Φ Rpprrfq) (where Φ It is L-naphthylalanine, R is D-arginine, P is D-proline), which is mainly used as a cyclic peptide inhibitor.
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Cat. No.: HY-168095
CAS No.: 3113279-03-8
Target:  

CXCR

Research Areas:  

Cancer

CXCR4 antagonist 10 (compound 21) is a potent antagonist of CXCR4, with the IC50 of 7.8 nM. CXCR4 antagonist 10 plays an important role in cancer research .
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Cat. No.: HY-P10200
CAS No.: 3032621-32-9
Target:  

Bacterial

Research Areas:  

Infection

CP7-FP13-2 is a peptide with antivirulence factor and antibacterial activity. CP7-FP13-2 inhibits the formation of Staphylococcus aureus biofilm and has good antibacterial efficacy in mice .
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Cat. No.: HY-P11432
Target:  

Melanocortin Receptor

Research Areas:  

Neurological Disease

PG-911 is a full MC5R agonist (EC50 = 0.031 nM for hMC5R). PG-911 is also a full antagonist at the hMC3R and the hMC4R (Kb: 0.38 nM and 0.17 nM, respectively). PG-911 can be used in the research of neurological disorders .
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Cat. No.: HY-P11469
CAS No.: 322639-20-3
PG-901 is a full, selective MC5R agonist (EC50 = 0.072 nM for hMC5R). PG-901 is also a full antagonist at the hMC3R and the hMC4R (Kb: 1.0 nM and 0.53 nM, respectively). PG-901 significantly diminishes Cytokines (IL-1α, IL-1β, IL-6). PG-901 increases glucose tolerance, reduces blood glucose, decreases retinal damage .
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Cat. No.: HY-P11912
Research Areas:  

Neurological Disease

Cyclo (Val-Val-Ile-d-Ala-Trp (Bodipy)-Gly) is a cyclic peptide-BODIPY conjugate. Cyclo (Val-Val-Ile-d-Ala-Trp (Bodipy)-Gly) detects prefibrillar 1-42 aggregates in neuronal cells, generating perinuclear punctate fluorescent spots. Cyclo (Val-Val-Ile-d-Ala-Trp (Bodipy)-Gly) is applicable to Alzheimer's disease-related research .
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Cat. No.: HY-P4992
CAS No.: 496849-46-8
Target:  

Somatostatin Receptor

Research Areas:  

Cancer

Tyr-(D-Dab4,Arg5,D-Trp8)-cyclo-Somatostatin-14 (4-11) is a somatostatin agonist that can be used in cancer research .
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Cat. No.: HY-P5738
CAS No.: 331714-57-9
Target:  

Bacterial

Research Areas:  

Infection

Palicourein is a 37 amino acid cyclic polypeptide. Palicourein inhibits the in vitro cytopathic effects of HIV-1RF infection of CEM-SS cells with an EC50 value of 0.1 μM and an IC50 value of 1.5 μM .
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Cat. No.: HY-P5739
CAS No.: 1803183-45-0
Target:  

Bacterial

Research Areas:  

Infection

Mram 8 is a cyclotide isolated from Viola philippica, a plant from the Violaceae family .
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Cat. No.: HY-P5753
CAS No.: 1873323-60-4
Target:  

Bacterial

Research Areas:  

Infection

JB-95, a β-hairpin macrocyclic peptide, exhibits potent antimicrobial activity against Escherichia coli. JB-95 can selectively disrupt the outer membrane but not the inner membrane of E. coli .
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Cat. No.: HY-P5753A
Target:  

Bacterial

Research Areas:  

Infection

JB-95 acetate, a β-hairpin macrocyclic peptide, exhibits potent antimicrobial activity against Escherichia coli. JB-95 acetate can selectively disrupt the outer membrane but not the inner membrane of E. coli .
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