2 Results for "

GTS21

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "GTS21" in MCE Product Catalog:

16
16 Cited Publications
Cat. No.: HY-14564A
CAS No.: 156223-05-1
Purity:  99.65%
Synonyms: DMXB-A; DMBX-anabaseine
Target:  

nAChR 5-HT Receptor

Research Areas:  

Inflammation/Immunology

GTS-21 dihydrochloride is a selective alpha7 nicotinic acetylcholine receptor (α7-nAChR) agonist with anti inflammatory and cognition enhancing activities. GTS-21 dihydrochloride is also a α4β2 (Ki=20 nM for humanα4β2) and 5-HT3A receptor (IC50=3.1 μM) antagonist .
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Cat. No.: HY-14564
CAS No.: 148372-04-7
Target:  

nAChR 5-HT Receptor

Research Areas:  

Inflammation/Immunology

GTS-21 dihydrochloride is a selective alpha7 nicotinic acetylcholine receptor (α7-nAChR) agonist with anti inflammatory and cognition enhancing activities. GTS-21 dihydrochloride is also a α4β2 (Ki=20 nM for humanα4β2) and 5-HT3A receptor (IC50=3.1 μM) antagonist. GTS-21 can be used in age-associated memory impairment (AAMI) and Alzheimer's disease research .
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