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42 Results for "
Sodium Channel inhibitor-1
" in MedChemExpress (MCE) Product Catalog:
Products (42)
42 Results for "Sodium Channel inhibitor-1" in MCE Product Catalog:
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Research Areas:
Sodium Channel inhibitor 1 is a state-dependent voltage-gated NaV1.7 inhibitor with an IC50 of 0.087 μM. Sodium Channel inhibitor 1 can be used for research of pain .
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91
91 Publications Verification
Synonyms: Sodium ascorbate; Sodium L-ascorbate; Vitamin C Sodium salt
6
6 Cited Publications
Synonyms: Endovion; NS3728
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Endovion is a pharmacological anion channel inhibitor (like chloride channel) and the specific VRAC/VSOAC blocker. Endovion (NS3728) is also an Anoctamin-1 (ANO 1) channel inhibitor .
4
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Dibucaine hydrochloride (Cinchocaine hydrochloride) is a sodium channel inhibitor. Dibucaine hydrochloride is a potent SChE inhibitor .
4
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Dibucaine (Cinchocaine) is a sodium channel inhibitor. Dibucaine is a potent SChE inhibitor .
2
2 Cited Publications
Synonyms: L-Ascorbate (Standard); Vitamin C (Standard)
2
2 Cited Publications
Synonyms: (±)-Norverapamil hydrochloride; D591 hydrochloride
Research Areas:
Norverapamil hydrochloride ((±)-Norverapamil hydrochloride), an N-demethylated metabolite of Verapamil, is a L-type calcium channel blocker and a P-glycoprotein (P-gp) function inhibitor .
Cat. No.: HY-B0166S
CAS No.: 1354064-87-1
Synonyms: L-Ascorbate-13C6; Vitamin C-13C6
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NaV1.7 inhibitor-1 is an efficacious voltage-gated sodium channel (NaV) 1.7 inhibitor with an IC50 of 0.6 nM for hNaV1.7, exhibits 80-fold selectivity versus hNaV1.5 .
Cat. No.: HY-B0166S1
CAS No.: 178101-88-7
Synonyms: L-Ascorbate-13C; Vitamin C-13C
Cat. No.: HY-44153
CAS No.: 689297-68-5
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KV2 channel inhibitor-1 is a selective KV2 channel inhibitor with IC50s of 0.2 μM and 0.41 μM for KV2.1 and KV2.2, respectively. KV2 channel inhibitor-1 possesses good selectivity over KV1.2 (IC50>10 μM). KV2 channel inhibitor-1 is >10-fold selective over NaV channels and other KV channels and displays weak activity on CaV channels .
Cat. No.: HY-155058
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Nav1.3 channel inhibitor 1 (compound 15b) is a state-dependent voltage-gated sodium channel Nav1.3 inhibitor (IC50=20 nM). Nav1.3 channel inhibitor 1 can penetrate the blood-brain barrier and can be used in the research of nervous system diseases .
Synonyms: NSC-609249 hydrochloride
Research Areas:
NSC-609249 hydrochloride is an impurity of Verapamil (HY-14275). Verapamil is a calcium channel blocker and a potent and orally active first-generation P-glycoprotein (P-gp) inhibitor .
Cat. No.: HY-122158
CAS No.: 903591-53-7
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CRAC channel inhibitor-1 (compound 55) is a CRAC channel inhibitor. CRAC channel inhibitor-1 can be used in immunology-related research .
Cat. No.: HY-P5818
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Cat. No.: HY-Z7760
CAS No.: 91189-59-2
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Felodipine 3,5-Dimethyl Ester is a aryldihydropyridine derivatives for use as mineralocorticoid receptor modulator and voltage-dependent L-type calcium channel CaV1.2 inhibitor .
Cat. No.: HY-101238S
CAS No.: 909556-32-7
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