85-79-0
Chemical Structure
Dibucaine
Synonym(s): Cinchocaine
- CAS No.: 85-79-0
- Formula:C20H29N3O2
- Molecular Weight:343.46
IUPAC Name: 2-butoxy-N-(2-(diethylamino)ethyl)quinoline-4-carboxamide
InChIKey: PUFQVTATUTYEAL-UHFFFAOYSA-N
SMILES: O=C(C1=CC(OCCCC)=NC2=CC=CC=C12)NCCN(CC)CC
Biological Activity: Dibucaine (Cinchocaine) is a sodium channel inhibitor. Dibucaine is a potent SChE inhibitor[1][2].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
Dibucaine | 99.69% | Dibucaine (Cinchocaine) is a sodium channel inhibitor. Dibucaine is a potent SChE inhibitor. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
Dibucaine (Standard) | ≥98% | Dibucaine (Standard) is the analytical standard of Dibucaine. This product is intended for research and analytical applications. Dibucaine (Cinchocaine) is a sodium channel inhibitor. Dibucaine is a potent SChE inhibitor. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
Dibucaine-d9 | Dibucaine-d9 is the deuterium labeled Dibucaine(HY-B0552).Dibucaine (Cinchocaine) is a sodium channel inhibitor. Dibucaine is a potent SChE inhibitor. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
Alloclamide | Alloclamide is a competitive antihistamine compound targeting the H1 histamine receptor. Alloclamide‘s core regulatory mechanism involves competitive binding to the H1 histamine receptor, blocking the activation of the receptor by histamine molecules and inhibiting various allergy-related biological responses mediated by histamine. Alloclamide can be used in allergy-related research. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
Viral 2C protein inhibitor 1 | Viral 2C protein inhibitor 1 (compound 6aw) is a potent and broad-spectrum enterovirus antiviral agent, inhibiting viral 2C protein. Viral 2C protein inhibitor 1 inhibits multiple strains of EV-D68, EV-A71 and CVB3 with EC50s of 0.1~3.6 µM, and exhibits high selectivity index and relatively low cytotoxicity. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
DKFZ-748 | 98.98% | DKFZ-748 is a selective HDAC10 inhibitor (pIC50=7.66), and shows anti-tumor activity. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
N-(2-(Diethylamino)ethyl)-2-iodobenzamide | N-(2-(Diethylamino)ethyl)-2-iodobenzamide can be radiolabeled and used for melanoma imaging. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
6-Amino-N-(2-(diethylamino)ethyl)quinoline-2-carboxamide | 99.67% | 6-Amino-N-(2-(diethylamino)ethyl)quinoline-2-carboxamide is a drug intermediate for synthesis of various active compounds. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
Dibucaine hydrochloride | 99.88% | Dibucaine hydrochloride (Cinchocaine hydrochloride) is a sodium channel inhibitor. Dibucaine hydrochloride is a potent SChE inhibitor. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
Bunaftide | Bunaftide (Bunaftine; Bunaphtide; Meregon) is an antiarrhythmic agent. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
2-Chloro-N-(2-(diethylamino)ethyl)quinoline-4-carboxamide (Standard) | ≥98% | 2-Chloro-N-(2-(diethylamino)ethyl)quinoline-4-carboxamide (Standard) is the analytical standard of 2-Chloro-N-(2-(diethylamino)ethyl)quinoline-4-carboxamide. This product is intended for research and analytical applications. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
Dibucaine-d9 hydrochloride | Dibucaine-d9 hydrochloride (Cinchocaine-d9 hydrochloride) is the deuterium labeled Dibucaine hydrochloride (HY-B0552A). Dibucaine hydrochloride (Cinchocaine hydrochloride) is a sodium channel inhibitor. Dibucaine hydrochloride is a potent SChE inhibitor. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
- [1]. Souto-Padron, T., A.P. Lima, and O. Ribeiro Rde, Effects of dibucaine on the endocytic/exocytic pathways in Trypanosoma cruzi. Parasitol Res, 2006. 99(4): p. 317-20. [Content Brief]
- [2]. Elamin, B., Dibucaine inhibition of serum cholinesterase. J Biochem Mol Biol, 2003. 36(2): p. 149-53. [Content Brief]