1 Result for "

VPC-3033

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "VPC-3033" in MCE Product Catalog:

Cat. No.: HY-118409
CAS No.: 110763-24-1
Target:  

Androgen Receptor

Research Areas:  

Endocrinology Cancer

VPC-3033 is an androgen receptor antagonist. VPC-3033 has a strong androgen DHT replacement potency (IC50: 0.625-2.5 μM), can effectively inhibit androgen receptor transcriptional activity (IC50=0.3 μM), and has a strong androgen receptor degradation ability. In addition, VPC-3033 exhibits significant anti-androgen receptor activity against prostate cancer cells resistant to Enzalutamide (HY-70002) .
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