4 Results for "

human monocytic U937 cells

" in MedChemExpress (MCE) Product Catalog:
Products (4)

4 Results for "human monocytic U937 cells" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-111449
CAS No.: 2162982-11-6
Purity:  99.78%
Synonyms: AHR antagonist 1
Research Areas:  

Inflammation/Immunology Cancer

BAY-218 (AHR antagonist 1) is an aryl hydrocarbon receptor (AHR) antagonist. BAY-218 has AHR inhibitory activity with an IC50 of 39.9 nM in in U87 glioblastoma cells. BAY-218 can be used for the research of cancer or conditions with dysregulated immune responses .
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Cat. No.: HY-162237
Target:  

RIP kinase

Research Areas:  

Inflammation/Immunology

RIPK1-IN-13 (compound 28) is a selective inhibitor for receptor-interacting serine/threonine-protein kinase 1 (RIPK1), the inhibitory activity is measured by ADP-Glo Kinase Assay with a pKi of 7.66. RIPK1-IN-13 inhibits human leukaemia cells U937 with a pIC50 of 7.2 .
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Cat. No.: HY-111449R
CAS No.: 2162982-11-6
Synonyms: AHR antagonist 1 (Standard)
BAY-218 (Standard) is the analytical standard of BAY-218 (HY-111449). This product is intended for research and analytical applications. BAY-218 (AHR antagonist 1) is an aryl hydrocarbon receptor (AHR) antagonist. BAY-218 has AHR inhibitory activity with an IC50 of 39.9 nM in in U87 glioblastoma cells. BAY-218 can be used for the research of cancer or conditions with dysregulated immune responses .
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Cat. No.: HY-N11852
CAS No.: 51415-08-8
Momilactone B is an inhibitor of α-amylase and α-glucosidase, with an IC50 of 146.85 μg/mL against Aspergillus oryzae α-amylase and an IC50 of 612.03 μg/mL against Saccharomyces cerevisiae α-glucosidase. Momilactone B upregulates the expression of p21 Waf1/Cip1, reduces the kinase activity of Cdk4 and Cdk6, induces cell cycle arrest and apoptosis in cancer cells, and triggers irreversible cell death via cell membrane damage. Momilactone B inhibits the growth of neighboring plant species and serves as a major contributing factor to the allelopathy of rice. Momilactone B can be used in studies related to rice allelopathy, type 2 diabetes, colon cancer and leukemia .
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