1. Signaling Pathways
  2. GPCR/G Protein
    Immunology/Inflammation
  3. CCR
  4. CCR2 Inhibitors

CCR2 Inhibitors

CCR1

CCR2

CCR3

CCR4

CCR5

CCR6

CCR7

CCR8

CCR9

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform CCR2 together.

Please try each isoform separately.

CCR2 Specific Antagonists
Product Name CCR2 CCR1 CCR5 CCR2 Selectivity Purity
RS 504393
CCR2, IC50: 89 nM
    Selective Antagonist 99.18%
PF-4136309
Human CCR2, IC50: 5.2 nM
Mouse CCR2, IC50: 13 nM
Rat CCR2, IC50: 17 nM
    Selective Antagonist 99.59%
RS102895 hydrochloride
CCR2, IC50: 360 nM
CCR1, IC50: 17800 nM
  Selective Antagonist 99.69%
TAK-779
MCP-1-CCR2b, IC50: 27 nM (in CHO/CCR5 cells)
 
MIP-1β-CCR5, IC50: 1 nM (in CHO/CCR5 cells)
RANTES-CCR5, IC50: 1.4 nM (in CHO/CCR5 cells)
MIP-1α-CCR5, IC50: 1 nM (in CHO/CCR5 cells)
Selective Antagonist 99.73%
MK-0812 Succinate
CCR2
    Selective Antagonist 99.69%
INCB 3284
MCP-1-hCCR2, IC50: 3.7 nM
    Selective Antagonist 99.30%
CCR2-RA-[R]
CCR2, IC50: 103 nM (in U2OS-CCR2 cells)
    Selective Antagonist 99.36%
MK-0812
CCR2
    Selective Antagonist 99.75%
Teijin compound 1
MCP-1-CCR2b, IC50: 180 nM
    Selective Antagonist 99.89%
CCR2 antagonist 1
CCR2, Ki: 2.4 nM
    Selective Antagonist
CCR2 antagonist 3
CCR2
    Selective Antagonist
RS102895
CCR2, IC50: 360 nM
CCR1, IC50: 17800 nM
  Selective Antagonist
Cenicriviroc
CCR2, IC50: 5.9 nM
 
CCR5, IC50: 0.29 nM
Pan Antagonist 98.07%
Cenicriviroc Mesylate
CCR2, IC50: 5.9 nM
 
CCR5, IC50: 0.29 nM
Pan Antagonist 98.58%
BMS-813160
CCR2
 
CCR5
Pan Antagonist 99.81%