1. Signaling Pathways
  2. GPCR/G Protein
    Immunology/Inflammation
  3. CCR
  4. CCR5 Inhibitors

CCR5 Inhibitors

CCR1

CCR2

CCR3

CCR4

CCR5

CCR6

CCR7

CCR8

CCR9

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform CCR5 together.

Please try each isoform separately.

CCR5 Specific Inhibitors & Antagonists
Product Name CCR5 CCR2 CCR5 Selectivity Purity
Cenicriviroc
CCR5, IC50: 0.29 nM
CCR2, IC50: 5.9 nM
Selective Antagonist 98.07%
Maraviroc
MIP-1α-CCR5, IC50: 3.3 nM (in HEK-293 cell membrane)
MIP-1β-CCR5, IC50: 7.2 nM (in HEK-293 cell membrane)
RANTES-CCR5, IC50: 5.2 nM (in HEK-293 cell membrane)
  Selective Antagonist 99.71%
Cenicriviroc Mesylate
CCR5, IC50: 0.29 nM
CCR2, IC50: 5.9 nM
Selective Antagonist 98.58%
TAK-779
MIP-1β-CCR5, IC50: 1 nM (in CHO/CCR5 cells)
RANTES-CCR5, IC50: 1.4 nM (in CHO/CCR5 cells)
MIP-1α-CCR5, IC50: 1 nM (in CHO/CCR5 cells)
MCP-1-CCR2b, IC50: 27 nM (in CHO/CCR5 cells)
Selective Antagonist 99.73%
DAPTA
gp120BaL/sCD4-CCR5, IC50: 55 pM (in Cf2Th/synR5 cells)
gp120CMCM235/sCD4-CCR5, IC50: 0.32 nM (in Cf2Th/synR5 cells)
  Selective Inhibitor 98.73%
Aplaviroc
CCR5
  Selective Antagonist
CCR5 antagonist 1
CCR5
  Selective Antagonist
BMS-813160
CCR5
CCR2
Pan Antagonist 99.81%