1. Signaling Pathways
  2. GPCR/G Protein
    Immunology/Inflammation
  3. CXCR
  4. CXCR3 Inhibitors

CXCR3 Inhibitors

CXCR

CXCR1

CXCR2

CXCR3

CXCR4

CXCR7

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform CXCR3 together.

Please try each isoform separately.

CXCR3 Specific Inhibitors, Agonists & Antagonists
Product Name CXCR3 CXCR3 Selectivity Purity
AMG 487
125I-IP10-CXCR3, IC50: 8 nM
125I-ITAC-CXCR3, IC50: 8.2 nM
Selective Inhibitor 99.65%
PS372424 hydrochloride
Human CXCR3
Selective Agonist >98.0%
SCH 546738
Human CXCR3, Ki: 0.4 nM
Selective Antagonist 99.23%
TAK-779
mCXCR3, IC50: 369 nM (in PBMCs)
Selective Antagonist 99.73%
NBI-74330
[125I]CXCL10-CXCR3, Ki: 1.5 nM (in CXCR3-CHO cell membranes)
[125I]CXCL11-CXCR3, Ki: 3.2 nM (in CXCR3-CHO cell membranes)
Selective Antagonist 99.23%
PS372424
Human CXCR3
Selective Agonist
AMG 487 (S-enantiomer)
CXCR3
Selective Antagonist 98.92%