DNA Methyltransferase Inhibitors

DNA Methyltransferase

DNMT1

DNMT3

MGMT

DNA Methyltransferase Inhibitors

Product Name	DNA Methyltransferase	DNMT1	DNMT3	MGMT	Purity
Decitabine		DNMT1	DNMT3A DNMT3B		99.97%
5-Azacytidine		DNMT1			99.79%
GSK-3484862		DNMT1			99.62%
RG108		CpG methylase M.SssI, IC₅₀: 115 nM			99.85%
5-Aza-4'-thio-2'-deoxycytidine		DNMT1
SGI-1027		DNMT1, IC₅₀: 12.5 μM	DNMT3B, IC₅₀: 7.5 μM DNMT3A, IC₅₀: 8 μM		99.77%
Hinokitiol		DNMT1			98.97%
CM-272		DNMT1, IC₅₀: 382 nM	DNMT3A, IC₅₀: 85 nM DNMT3B, IC₅₀: 1200 nM		99.27%
Zebularine		DNMT1	DNMT3a/3L		99.99%
γ-Oryzanol		DNMT1, IC₅₀: 3.2 μM	DNMT3A, IC₅₀: 22.3 μM
Guadecitabine sodium		DNMT1			98.05%
DNMT3A-IN-1			DNMT3A		98.81%
Lomeguatrib				MGMT, IC₅₀: 9 nM MGMT, IC₅₀: 6 nM (in MCF-7 cells)	99.70%
DY-46-2			DNMT3A, IC₅₀: 0.39 μM		99.32%
CM-579 trihydrochloride	DNA Methyltransferase, IC₅₀: 32 nM	DNMT1, Kd: 1.5 nM	DNMT3A, IC₅₀: 92 nM DNMT3B, IC₅₀: 1000 nM		98.03%
DC_517		DNMT1, Kd: 0.91 μM DNMT1, IC₅₀: 1.7 μM			99.41%
(R)-GSK-3685032		DNMT1			98.02%
O6BTG-octylglucoside				MGMT, IC₅₀: 32 nM
DC-05		DNMT1, Kd: 1.09 μM DNMT1, IC₅₀: 10.3 μM			99.08%
Guadecitabine	DNA Methyltransferase				98.0%
CM-579	DNA Methyltransferase, IC₅₀: 32 nM	DNMT1, Kd: 1.5 nM	DNMT3A, IC₅₀: 92 nM DNMT3B, IC₅₀: 1000 nM
Nanaomycin A			DNMT3B, IC₅₀: 500 nM		98.18%
Isofistularin-3		DNMT1, IC₅₀: 13.5 μM
(4aS,8aR)-NPD-001			DNMT3A
DNMT-IN-1	DNA Methyltransferase, EC₅₀: 3.2 μM

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