1. Signaling Pathways
  2. Cell Cycle/DNA Damage
    Cytoskeleton
  3. Kinesin
  4. Kinesin Inhibitors

Kinesin Inhibitors

Kinesin-5/Eg5/KSP

Kinesin-6

Kinesin-7/CENP-E

Kinesin-12

Kinesin-14

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Kinesin Inhibitors
Product Name Kinesin-5/Eg5/KSP Kinesin-6 Kinesin-7/CENP-E Kinesin-12 Kinesin-14 Purity
Ispinesib
KSP, Ki app: 1.7 nM
        99.62%
Filanesib
KSP, IC50: 6 nM
        99.59%
GSK-923295    
CENP-E, Ki: 1.6 nM (Canine CENP-E)
    99.82%
AZ82        
HSET/KIFC1, IC50: 300 nM
HSET/KIFC1, Ki: 43 nM
99.31%
Monastrol
Eg5, IC50: 14 μM
        99.70%
Litronesib
Eg5
        99.59%
SB-743921 hydrochloride
Eg5, Ki: 0.1 nM
        99.87%
S-Trityl-L-cysteine
Eg5
        98.99%
Paprotrain  
MKLP-2, IC50: 1.35 μM
      99.87%
EMD534085
Kinesin-5, IC50: 8 nM
        99.55%
Kif15-IN-1      
KIF15
  99.39%
CW-069        
HSET, IC50: 75 μM
98.99%
Dimethylenastron
Eg5, IC50: 200 nM
        98.68%
PF-2771    
CENP-E, IC50: 16.1 nM
    99.76%
K858 (Racemic)
Eg5, IC50: 1.3 μM
        99.83%
ARQ 621
Eg5
        ≥99.0%
PVZB1194
Eg5
        99.90%
Kif15-IN-2      
KIF15
  98.64%
MK-0731
KSP, IC50: 2.2 nM
       
Eg5 Inhibitor V, trans-24
Eg5, IC50: 0.65 μM