1. シグナル伝達
  2. Metabolic Enzyme/Protease
  3. NADPH Oxidase
  4. NADPH Oxidase Inhibitors

NADPH Oxidase Inhibitors

NOX1

NOX2

NOX4

NOX5

DUOX1

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

NADPH Oxidase Inhibitors
製品名 NOX1 NOX2 NOX4 NOX5 DUOX1 純度
GSK2795039  
NOX2
      98.56%
Setanaxib
NOX1
 
NOX4
    99.81%
CPP11G  
NOX2, IC50: 20 μM
     
GK-136901
NOX1, Ki: 160 nM
 
NOX4, Ki: 165 nM
   
GLX351322    
NOX4
    99.48%
ML171
NOX1
        99.53%
APX-115
NOX1
NOX2
NOX4
    99.90%
Prochlorperazine dimaleate
NOX1, : 6.4 μM
NOX2, : 4.5 μM
 
NOX5, : 2.3 μM
  ≥98.0%
GKT136901
NOX1
 
NOX4
    99.70%
NoxA1ds
NOX1
       
APX-115 free base
NOX1
NOX2
NOX4
    99.54%
NADPH oxidase-IN-1  
NOX2, IC50: 1.9 μM
NOX4, IC50: 2.47 μM
    99.69%
Mulberrofuran G    
NOX4
   
Fluoflavine
NOX1
        98.47%
NCATS-SM7270  
NOX2, IC50: 4.09 μM
      99.17%
Hidrosmin
NOX1
 
NOX4
   
(Rac)-Nebivolol  
NOX2
     
MC4762  
NOX2, IC50: 0.155 μM
     
NoxA1ds TFA
NOX1
       
Niazirin    
NOX4
    99.9%
NOX5-IN-1
NOX1, IC50: >100 μM
NOX2, IC50: >100 μM
NOX4, IC50: >100 μM
NOX5, IC50: 0.3 μM
DUOX1, IC50: >15 μM
NOX5-IN-2
NOX1, IC50: >100 μM
NOX2, IC50: >100 μM
NOX4, IC50: >100 μM
NOX5, IC50: 0.70 μM
DUOX1, IC50: >15 μM
AMPAR modulator-12
NOX1
       
GLX481372
NOX1, IC50: 7 μM
NOX2, IC50: 16 μM
NOX4, IC50: 0.68 μM
NOX5, IC50: 0.57 μM
 
ML171 analog 1
NOX1