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Cat. No.: HY-175790

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AR/BET ligand-1

AR/BET ligand-1 is a AR/BET ligand, which can be used for the synthesis of PROTACs, such as PROTAC AR/BET protein degrader-1 (HY-160262).

For research use only. We do not sell to patients.

CAS No.: 2493425-86-6
Formula: C₂₂H₂₁N₃O
Molecular Weight:343.42

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

AR/BET ligand-1 Chemical Structure

CAS No.: 2493425-86-6

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
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Description

AR/BET ligand-1 is a AR/BET ligand, which can be used for the synthesis of PROTACs, such as PROTAC AR/BET protein degrader-1 (HY-160262)^[1].

IC₅₀ & Target^[1]

BET

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Chemical Information

CAS No. 2493425-86-6
Molecular Weight 343.42
Formula C₂₂H₂₁N₃O
SMILES

CC1=NOC(C)=C1C2=CC=C(C)C(NC3=CC=C(C4(C#N)CC4)C=C3)=C2
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Lyu Haibin, et al. Aromatic Amine Ar and Bet Targeted Protein Degradation Chimeric Compound and Application Thereof. CN-111944012-A

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References

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AR/BET ligand-1

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AR/BET ligand-1 Related Classifications

HY-175790 Related Classifications