Bromodomain inhibitor-10
Bromodomain inhibitor-10 (compound 128) is a potent bromodomain inhibitor with Kds of 15.0, 2500 nM for BRD4-1 and BRD4-2, respectively. Bromodomain inhibitor-10 inhibits the production of IL12p40.
For research use only. We do not sell to patients.
- CAS No.: 1870849-58-3
- Formula: C20H20N4O3
- Molecular Weight:364.40
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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BRD4-1 15 nM (Kd) |
BRD4-2 2500 nM (Kd) |
Chemical Information
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CAS No. 1870849-58-3
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Molecular Weight 364.40
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Formula C20H20N4O3
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SMILES
CC1=CC(NC2=C1C=C(NC(C3=C(N4CCOCC4)N=CC=C3)=O)C=C2)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)