country

Change Language

EN - English
FR - Français
DE - Deutsch
ES - Español
JA - 日本語
KO - 한국어

Country or Region:

United States

Product Name	Size / Unit Price	Qty

Total: USD 0.00 Checkout

Cat. No.: HY-184400

Copy Link Print Information

Pynazolam

Pynazolam is a predicted positive allosteric modulator of GABA_A receptor. 3D-field QSAR and RVM models predict an IC₅₀ of approximately 0.40 nM. Pynazolam can be used in studies related to GABA_A receptor pharmacology.

Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.

CAS No.: 2034366-97-5
Formule: C₁₆H₁₂N₆O₂
Masse moléculaire:320.31

Stockage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Pynazolam Chemical Structure

CAS No.: 2034366-97-5

Stock

Quantité

Amount: USD 0.00

* Veuillez sélectionner la quantité avant d'ajouter des articles.

Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
- In Vitro
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
Bioz

Activité biologique

Description

IC₅₀ & Target

^[1]

GABA_A receptor

In Vitro

Pynazolam is predicted to be one of the most active designer benzodiazepines at the GABA-AR, with a log 1/c value of 9.4, indicating potent inhibitory activity in displacing [³H]-diazepam from rat cerebral cortex binding sites^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 2034366-97-5
Masse moléculaire 320.31
Formule C₁₆H₁₂N₆O₂
SMILES

O=[N+](C1=CC=C(N2C(CN=C3C4=NC=CC=C4)=NN=C2C)C3=C1)[O-]
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Instruction de manipulation (2659 KB)

Références

[1]. Catalani V, et al. In silico studies on recreational drugs: 3D quantitative structure activity relationship prediction of classified and de novo designer benzodiazepines. Chemical biology & drug design. 2023 Jan;101(1):40-51. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

Keywords

MOQ

Minimum order quantity

100 mg

Obtenir un devis En stock

Other size

Obtenir un devis