102636-74-8
102636-74-8
Chemical Structure
CINPA1
- CAS No.: 102636-74-8
- Formula:C23H29N3O3
- Molecular Weight:395.49
IUPAC Name: ethyl (5-(diethylglycyl)-10,11-dihydro-5H-dibenzo[b,f]azepin-3-yl)carbamate
InChIKey: AYQBYSPEGRYKFA-UHFFFAOYSA-N
SMILES: CCN(CC)CC(N1C2=CC(NC(OCC)=O)=CC=C2CCC3=C1C=CC=C3)=O
Biological Activity: CINPA1 is a potent and specific inhibitor of constitutive androstane receptor (CAR) that does not activate pregnane X receptor (PXR). CINPA1 reduces CAR-mediated transcription with an IC50 of ~70 nM. CINPA1 can be used as a molecular tool for understanding CAR function[1].
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CINPA1 | 99.80% | CINPA1 is a potent and specific inhibitor of constitutive androstane receptor (CAR) that does not activate pregnane X receptor (PXR). CINPA1 reduces CAR-mediated transcription with an IC50 of ~70 nM. CINPA1 can be used as a molecular tool for understanding CAR function. | ||||||||||||||||||||
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References
Keywords
