1170321-92-2
Chemical Structure
ELOVL6-IN-4
- CAS No.: 1170321-92-2
- Formula:C20H20F3N3O3S
- Molecular Weight:439.45
IUPAC Name: (1R,3r,5S)-3-(pyridin-2-ylsulfonyl)-N-(4-(trifluoromethyl)phenyl)-8-azabicyclo[3.2.1]octane-8-carboxamide
InChIKey: WYCGDOXAJCYGEC-FVQHAEBGSA-N
SMILES: FC(F)(F)C(C=C1)=CC=C1NC(N2[C@@]3([H])C[C@@H](C[C@]2([H])CC3)S(=O)(C4=CC=CC=N4)=O)=O
Biological Activity: ELOVL6-IN-4 is a potent, selective, and orally active long chain fatty acid elongase 6 (ELOVL6) inhibitor with IC50s of 79 nM and 94 nM for human and mouse ELOVL6, respectively. ELOVL6-IN-4 shows excellent selectivity over the other human ELOVL subtypes (ELOVL1, -2, -3, and -5) and mouse ELOVL3[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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ELOVL6-IN-4 | 98.94% | ELOVL6-IN-4 is a potent, selective, and orally active long chain fatty acid elongase 6 (ELOVL6) inhibitor with IC50s of 79 nM and 94 nM for human and mouse ELOVL6, respectively. ELOVL6-IN-4 shows excellent selectivity over the other human ELOVL subtypes (ELOVL1, -2, -3, and -5) and mouse ELOVL3. | ||||||||||||||||||||
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Keywords
