1185003-32-0
1185003-32-0
Chemical Structure
PGK1-IN-3
- CAS No.: 1185003-32-0
- Formula:C18H17N3O4S2
- Molecular Weight:403.48
InChIKey: TUTZYYLPVTZWDA-UHFFFAOYSA-N
SMILES: O=C1NC2=C(C(NC3CCCCC3)=O)SC(N2C4=CC5=C(C=C14)OCO5)=S
Biological Activity: PGK1-IN-3 is an orally active PGK1 inhibitor with human PGK1 IC50 values of 0.48 μM and human PGK1 Kd of 63 nM. PGK1-IN-3 binds to the ADP-binding pocket of PGK1, inhibits glycolysis, and reduces glucose consumption and lactate production. PGK1-IN-3 can be used for the research of pancreatic cancer[1].
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PGK1-IN-3 | PGK1-IN-3 is an orally active PGK1 inhibitor with human PGK1 IC50 values of 0.48 μM and human PGK1 Kd of 63 nM. PGK1-IN-3 binds to the ADP-binding pocket of PGK1, inhibits glycolysis, and reduces glucose consumption and lactate production. PGK1-IN-3 can be used for the research of pancreatic cancer. | |||||||||||||||||||||
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