1197420-05-5
1197420-05-5
Chemical Structure
BMS-819881
- CAS No.: 1197420-05-5
- Formula:C24H21ClN2O4S
- Molecular Weight:468.95
IUPAC Name: (R)-6-(4-chlorophenyl)-3-(4-(2-cyclopropyl-2-hydroxyethoxy)-3-methoxyphenyl)thieno[3,2-d]pyrimidin-4(3H)-one
InChIKey: WKMOSCAIWUUQPD-IBGZPJMESA-N
SMILES: ClC1=CC=C(C2=CC(N=CN(C3=CC(OC)=C(OC[C@H](O)C4CC4)C=C3)C5=O)=C5S2)C=C1
Biological Activity: BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM. BMS-819881 also is selective and potent for CYP3A4 activity with an EC50 of 13 μM.
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BMS-819881 | 99.78% | BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM. BMS-819881 also is selective and potent for CYP3A4 activity with an EC50 of 13 μM. | ||||||||||||||||||||
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Keywords
