1262032-38-1
1262032-38-1
Chemical Structure
MeThPmR
- CAS 番号: 1262032-38-1
- Formula:C12H14N2O5S
- Molecular Weight:298.31
InChIKey: IHMAIWVMISBALC-TURQNECASA-N
SMILES: O=C1N([C@H]2[C@H](O)[C@H](O)[C@@H](CO)O2)C=C(C=C(C)S3)C3=N1
Biological Activity: MeThPmR, a ribonucleoside derivative, is a potent and selective human nucleoside transporter 1 (hCNT1) inhibitor (Ki/sub> = 0.16-0.69 μM). MeThPmR exhibit weak inhibitory activity on hCNT2 (IC50 = 360 μM) and hCNT3 (Ki = 4.7 μM). MeThPmR can protect cells from the toxicity of nucleoside drugs. MeThPmR can be used for the research of cancer[1].
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MeThPmR | MeThPmR, a ribonucleoside derivative, is a potent and selective human nucleoside transporter 1 (hCNT1) inhibitor (Ki/sub> = 0.16-0.69 μM). MeThPmR exhibit weak inhibitory activity on hCNT2 (IC50 = 360 μM) and hCNT3 (Ki = 4.7 μM). MeThPmR can protect cells from the toxicity of nucleoside drugs. MeThPmR can be used for the research of cancer. | |||||||||||||||||||||
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