130325-35-8
Chemical Structure
PD 135158
Synonym(s): CAM 1028
- CAS No.: 130325-35-8
- Formula:C42H61N5O11
- Molecular Weight:811.96
IUPAC Name: (2R,3R,4R,5S)-6-(methylamino)hexane-1,2,3,4,5-pentaol 4-(((R)-2-((R)-3-(1H-indol-3-yl)-2-methyl-2-(((((1S,2R,4S)-1,7,7-trimethylbicyclo[2.2.1]heptan-2-yl)oxy)carbonyl)amino)propanamido)-1-phenylethyl)amino)-4-oxobutanoate
InChIKey: CWJXTOIDFOBOKQ-OWZHFMFPSA-N
SMILES: C[C@@](C1(C)C)(CC[C@@]1([H])C2)[C@@H]2OC(N[C@](C(NC[C@@H](C3=CC=CC=C3)NC(CCC(O)=O)=O)=O)(C)CC4=CNC5=CC=CC=C45)=O.O[C@H]([C@@H](O)CNC)[C@H](O)[C@H](O)CO
Biological Activity: PD 135158 (CAM 1028) is a selective CCKB receptor antagonist with an IC50 of 2.8 nM against mouse cortex CCKB. PD 135158 shows anxiolytic activity[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PD 135158 | PD 135158 (CAM 1028) is a selective CCKB receptor antagonist with an IC50 of 2.8 nM against mouse cortex CCKB. PD 135158 shows anxiolytic activity. | |||||||||||||||||||||
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