1360053-81-1
1360053-81-1
Chemical Structure
Spebrutinib besylate
Synonym(s): AVL-292 benzenesulfonate; CC-292 besylate
- CAS No.: 1360053-81-1
- Formula:C28H28FN5O6S
- Molecular Weight:581.62
IUPAC Name: N-(3-((5-fluoro-2-((4-(2-methoxyethoxy)phenyl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide benzenesulfonate
InChIKey: ABSXPNGWJFAPRT-UHFFFAOYSA-N
SMILES: COCCOC1=CC=C(NC2=NC=C(F)C(NC3=CC=CC(NC(C=C)=O)=C3)=N2)C=C1.O=S(C4=CC=CC=C4)(O)=O
Biological Activity: Spebrutinib besylate (AVL-292 benzenesulfonate; CC-292 besylate) is a potent inhibitor of Btk kinase activity (IC50<0.5 nM, Kinact/Ki=7.69×104 M-1s-1s) in biochemical assays.
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Spebrutinib besylate | Spebrutinib besylate (AVL-292 benzenesulfonate; CC-292 besylate) is a potent inhibitor of Btk kinase activity (IC50<0.5 nM, Kinact/Ki=7.69×104 M-1s-1s) in biochemical assays. | |||||||||||||||||||||
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