149629-70-9
Chemical Structure
Impentamine dihydrobromide
Synonym(s): VUF 4702 dihydrobromide
- CAS No.: 149629-70-9
- Formula:C8H17Br2N3
- Molecular Weight:315.05
IUPAC Name: 5-(1H-imidazol-5-yl)pentan-1-amine dihydrobromide
InChIKey: QSDXAAWBBPWGEL-UHFFFAOYSA-N
SMILES: NCCCCCC1=CN=CN1.[H]Br.[H]Br
Biological Activity: Impentamine dihydrobromide (VUF 4702 dihydrobromide) is a histamine H3 receptor antagonist with potential antihistamine activity. Impentamine dihydrobromide shows the strongest selective H3 antagonism among a series of 4(5)-(ω-aminoalkyl)-1H-imidazole compounds. The pA2 value of impentamine dihydrobromide is 8.4, showing its high efficacy in guinea pig jejunum. Impentamine dihydrobromide has a specific antagonistic binding site with the H3 receptor[1].
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Impentamine dihydrobromide | Impentamine dihydrobromide (VUF 4702 dihydrobromide) is a histamine H3 receptor antagonist with potential antihistamine activity. Impentamine dihydrobromide shows the strongest selective H3 antagonism among a series of 4(5)-(ω-aminoalkyl)-1H-imidazole compounds. The pA2 value of impentamine dihydrobromide is 8.4, showing its high efficacy in guinea pig jejunum. Impentamine dihydrobromide has a specific antagonistic binding site with the H3 receptor. | |||||||||||||||||||||
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