174688-78-9

CH 275 Chemical Structure
174688-78-9

Chemical Structure

CH 275

  • CAS No.: 174688-78-9
  • Formula:C74H96N14O15S2
  • Molecular Weight:1485.77

IUPAC Name: (4R,7S,10S,13S,16S,19S,22R,25S,28S,31S,34R)-22-((1H-indol-3-yl)methyl)-34-amino-31-(4-aminobutyl)-13,25,28-tribenzyl-10,16-bis((R)-1-hydroxyethyl)-7-(hydroxymethyl)-19-(4-((isopropylamino)methyl)benzyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decaazacyclopentatriacontane-4-carboxylic acid

InChIKey: SYHQUPOPQRNSKD-SKMHOITNSA-N

SMILES: O=C(N[C@H](C(N[C@@](C(N[C@H](C(N[C@@](C(N[C@H](C(N1)=O)CO)=O)([H])[C@H](O)C)=O)CC2=CC=CC=C2)=O)([H])[C@H](O)C)=O)CC(C=C3)=CC=C3CNC(C)C)[C@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CSSC[C@H]1C(O)=O)N)=O)CCCCN)=O)CC4=CC=CC=C4)=O)CC5=CC=CC=C5)=O)CC6=CNC7=CC=CC=C67

Biological Activity: CH 275 is a peptide analog of somatostatin and binds preferably to somatostatin receptor 1 (sst1) with a Ki of 52 nM[1]. CH 275 acts as a potent and selective sst1 agonist (IC50=30.9 nM) and also displays IC50 values of 345 nM, >1 μM, >10 μM, >10 μM for human sst3, sst4, sst2 and sst5, respectively[2]. CH 275 can be used for the research of alzheimer’s disease[3].

Cat. No. Product Name Purity Description Pricing
HY-P1206 		CH 275 99.52% CH 275 is a peptide analog of somatostatin and binds preferably to somatostatin receptor 1 (sst1) with a Ki of 52 nM. CH 275 acts as a potent and selective sst1 agonist (IC50=30.9 nM) and also displays IC50 values of 345 nM, >1 μM, >10 μM, >10 μM for human sst3, sst4, sst2 and sst5, respectively. CH 275 can be used for the research of alzheimer’s disease.
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