1883545-52-5
Chemical Structure
MM-102 TFA
Synonym(s): HMTase Inhibitor IX TFA
- No. CAS: 1883545-52-5
- Formula:C37H50F5N7O6
- Molecular Weight:783.83
IUPAC Name: (S)-N-(bis(4-fluorophenyl)methyl)-1-(2-(2-ethyl-2-isobutyramidobutanamido)-5-guanidinopentanamido)cyclopentane-1-carboxamide 2,2,2-trifluoroacetate
InChIKey: ZRKTWBXVGMHWHM-YCBFMBTMSA-N
SMILES: O=C(C1(NC([C@@H](NC(C(NC(C(C)C)=O)(CC)CC)=O)CCCNC(N)=N)=O)CCCC1)NC(C2=CC=C(F)C=C2)C3=CC=C(F)C=C3.FC(F)(F)C(O)=O
Biological Activity: MM-102 TFA (HMTase Inhibitor IX TFA) is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM with an estimated Ki < 1 nM in WDR5 binding assay, which is >200 times more potent than the ARA peptide.
| Referencia número | Nombre del producto | Pureza | Descripciòn | Pricing | |||||||||||||||||||
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MM-102 TFA | 99.68% | MM-102 TFA (HMTase Inhibitor IX TFA) is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM with an estimated Ki < 1 nM in WDR5 binding assay, which is >200 times more potent than the ARA peptide. | ||||||||||||||||||||
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