2021249-10-3
Chemical Structure
Vilanterol-d4 trifenatate
Synonym(s): GW642444-d4 trifenatate
- CAS No.: 2021249-10-3
- Formula:C44H45D4Cl2NO7
- Molecular Weight:778.79
IUPAC Name: (R)-4-(2-((6-(2-((2,6-dichlorobenzyl)oxy)ethoxy-1,1,2,2-d4)hexyl)amino)-1-hydroxyethyl)-2-(hydroxymethyl)phenol 2,2,2-triphenylacetate
InChIKey: KLOLZALDXGTNQE-UCSYHREKSA-N
SMILES: OC(C(C1=CC=CC=C1)(C2=CC=CC=C2)C3=CC=CC=C3)=O.ClC(C=CC=C4Cl)=C4COC([2H])([2H])C([2H])([2H])OCCCCCCNC[C@@H](C5=CC(CO)=C(C=C5)O)O
Biological Activity: Vilanterol-d4 (trifenatate) is deuterium labeled Vilanterol (trifenatate).Vilanterol (GW642444) acetate is a long-acting β2 adrenergic receptor agonist. Vilanterol acetate has pEC50 values for β2-AR, β1-AR, and β3-AR of 9.4, 6.4, and 6.1, respectively. Vilanterol acetate selectively activates airway β2 adrenergic receptors, increases cAMP and thus relaxes bronchial smooth muscle. Vilanterol acetate can be used in asthma research.
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Vilanterol-d4 trifenatate | Vilanterol-d4 (trifenatate) is deuterium labeled Vilanterol (trifenatate).Vilanterol (GW642444) acetate is a long-acting β2 adrenergic receptor agonist. Vilanterol acetate has pEC50 values for β2-AR, β1-AR, and β3-AR of 9.4, 6.4, and 6.1, respectively. Vilanterol acetate selectively activates airway β2 adrenergic receptors, increases cAMP and thus relaxes bronchial smooth muscle. Vilanterol acetate can be used in asthma research. | |||||||||||||||||||||
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Vilanterol trifenatate | 99.82% | Vilanterol (GW642444) trifenatate is a long-acting β2 adrenergic receptor agonist. Vilanterol trifenatate has pEC50 values for β2-AR, β1-AR, and β3-AR of 9.4, 6.4, and 6.1, respectively. Vilanterol trifenatate selectively activates airway β2 adrenergic receptors, increases cAMP and thus relaxes bronchial smooth muscle. Vilanterol trifenatate can be used in asthma research. | ||||||||||||||||||||
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