2055397-28-7
2055397-28-7
Chemical Structure
WM-1119
- CAS No.: 2055397-28-7
- Formula:C18H13F2N3O3S
- Molecular Weight:389.38
IUPAC Name: 2-fluoro-N'-(3-fluoro-5-(pyridin-2-yl)benzoyl)benzenesulfonohydrazide
InChIKey: QLXULUNLCRKWRD-UHFFFAOYSA-N
SMILES: O=C(NNS(=O)(C1=CC=CC=C1F)=O)C2=CC(C3=NC=CC=C3)=CC(F)=C2
Biological Activity: WM-1119, a chemical probe, is a highly potent and selective KAT6A inhibitor, with an IC50 of 0.25 μM for KAT6A in lymphoma cells, the binding KD values of WM-1119 with KAT6A, KAT5 and KAT7 are 2 nM, 2.2 μM, 0.5 μM , respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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WM-1119 | 99.57% | WM-1119, a chemical probe, is a highly potent and selective KAT6A inhibitor, with an IC50 of 0.25 μM for KAT6A in lymphoma cells, the binding KD values of WM-1119 with KAT6A, KAT5 and KAT7 are 2 nM, 2.2 μM, 0.5 μM , respectively. | ||||||||||||||||||||
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WM-1119 (Standard) | ≥98% | WM-1119 (Standard) is the analytical standard of WM-1119 (HY-102058). This product is intended for research and analytical applications. WM-1119, a chemical probe, is a highly potent and selective KAT6A inhibitor, with an IC50 of 0.25 μM for KAT6A in lymphoma cells, the binding Kd values of WM-1119 with KAT6A, KAT5 and KAT7 are 2 nM, 2.2 μM, 0.5 μM , respectively. | ||||||||||||||||||||
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References
Keywords
