2101958-02-3
Chemical Structure
Squarunkin A
- CAS No.: 2101958-02-3
- Formula:C25H32F3N5O4
- Molecular Weight:523.55
IUPAC Name: ethyl 4-((3,4-dioxo-2-((2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl)amino)cyclobut-1-en-1-yl)amino)piperidine-1-carboxylate
InChIKey: ZKITWOVRRSBKFG-UHFFFAOYSA-N
SMILES: O=C(N1CCC(NC2=C(NCCN3CCN(C4=CC=CC(C(F)(F)F)=C4)CC3)C(C2=O)=O)CC1)OCC
Biological Activity: Squarunkin A is a potent and selective UNC119-cargo interaction inhibitor, interrupting the UNC119A-myristoylated Src N-terminal peptide interaction (IC50=10 nM). Squarunkin A interferes with the activation of Src kinase in cells[1].
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Squarunkin A | 99.49% | Squarunkin A is a potent and selective UNC119-cargo interaction inhibitor, interrupting the UNC119A-myristoylated Src N-terminal peptide interaction (IC50=10 nM). Squarunkin A interferes with the activation of Src kinase in cells. | ||||||||||||||||||||
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Keywords
