2170732-60-0
2170732-60-0
Chemical Structure
ERRγ-IN-1
- CAS No.: 2170732-60-0
- Formula:C30H36N2O2
- Molecular Weight:456.62
InChIKey: RUUIHSHMHGOGMZ-QVIHXGFCSA-N
SMILES: OCCC/C(C1=CC=CC=C1)=C(C2=CC=C(C=C2)O)/C3=CC=C(N4CCN(CC4)C(C)C)C=C3
Biological Activity: ERRγ-IN-1 is a ERRγ inhibitor with an IC50 of 0.040 μM. ERRγ-IN-1 activates MAPK (p44/p42) and inhibits the activity of ERRγ. ERRγ-IN-1 significantly increases iodine uptake in anaplastic thyroid carcinoma xenografts and suppresses tumor growth in nude mice. ERRγ-IN-1 is applicable for the research of anaplastic thyroid carcinoma[1].
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ERRγ-IN-1 | ERRγ-IN-1 is a ERRγ inhibitor with an IC50 of 0.040 μM. ERRγ-IN-1 activates MAPK (p44/p42) and inhibits the activity of ERRγ. ERRγ-IN-1 significantly increases iodine uptake in anaplastic thyroid carcinoma xenografts and suppresses tumor growth in nude mice. ERRγ-IN-1 is applicable for the research of anaplastic thyroid carcinoma. | |||||||||||||||||||||
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