2230880-25-6
2230880-25-6
Chemical Structure
Ar-V7-IN-1
- CAS No.: 2230880-25-6
- Formula:C10H10Br2N4OS
- Molecular Weight:394.09
IUPAC Name: L-lysine-13C6-15N2 hydrochloride
InChIKey: KEFGZKYLWGZFFS-UHFFFAOYSA-N
SMILES: BrC1=C(Br)N(C2=CSC(N3CCOCC3)=N2)C=N1
Biological Activity: Ar-V7-IN-1 is a potent inhibitor of Ar-V7. Ar-V7-IN-1 inhibits the transcriptional activity of androgen receptor (AR) and the secretion of prostate-specific antigen (PSA) with an eGFP IC50 of 1232 nM and the PSA IC50 of 1391 μM. Ar-V7-IN-1 has the potential for the research of various indications, in particular cancers such as prostate cancer[1].
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Ar-V7-IN-1 | 98.02% | Ar-V7-IN-1 is a potent inhibitor of Ar-V7. Ar-V7-IN-1 inhibits the transcriptional activity of androgen receptor (AR) and the secretion of prostate-specific antigen (PSA) with an eGFP IC50 of 1232 nM and the PSA IC50 of 1391 μM. Ar-V7-IN-1 has the potential for the research of various indications, in particular cancers such as prostate cancer. | ||||||||||||||||||||
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