2309668-44-6
2309668-44-6
Chemical Structure
Derazantinib Racemate
Synonym(s): ARQ-087 Racemate
- CAS No.: 2309668-44-6
- Formula:C29H29FN4O
- Molecular Weight:468.57
IUPAC Name: 6-(2-fluorophenyl)-N-(3-(2-((2-methoxyethyl)amino)ethyl)phenyl)-5,6-dihydrobenzo[h]quinazolin-2-amine
InChIKey: KPJDVVCDVBFRMU-UHFFFAOYSA-N
SMILES: COCCNCCC1=CC(NC2=NC=C3CC(C4=CC=CC=C4F)C5=CC=CC=C5C3=N2)=CC=C1
Biological Activity: Derazantinib Racemate (ARQ-087 Racemate) is the racemate of Derazantinib. Derazantinib is an orally bioavailable, ATP competitive tyrosine kinase inhibitor; exhibits potent activity against FGFR1-3 chondrocytes with IC50s of 4.5, 1.8, and 4.5 nM, respectively.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Derazantinib Racemate | 99.38% | Derazantinib Racemate (ARQ-087 Racemate) is the racemate of Derazantinib. Derazantinib is an orally bioavailable, ATP competitive tyrosine kinase inhibitor; exhibits potent activity against FGFR1-3 chondrocytes with IC50s of 4.5, 1.8, and 4.5 nM, respectively. | ||||||||||||||||||||
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