2377335-74-3
2377335-74-3
Chemical Structure
M-808
- CAS No.: 2377335-74-3
- Formula:C45H63FN6O5S
- Molecular Weight:819.08
IUPAC Name: methyl ((1S,2R)-2-((S)-2-(azetidin-1-yl)-1-(3-fluorophenyl)-1-(1-((1-(4-((1-((E)-4-(piperidin-1-yl)but-2-enoyl)azetidin-3-yl)sulfonyl)phenyl)azetidin-3-yl)methyl)piperidin-4-yl)ethyl)cyclopentyl)carbamate
InChIKey: BTSUNSRQYLVGIS-ADTYUTHVSA-N
SMILES: O=S(C(C=C1)=CC=C1N(C2)CC2CN(CC3)CCC3[C@@]([C@@]4([H])CCC[C@@H]4NC(OC)=O)(CN5CCC5)C6=CC(F)=CC=C6)(C7CN(C(/C=C/CN8CCCCC8)=O)C7)=O
Biological Activity: M-808 is a highly potent and efficacious covalent Menin-MLL interaction inhibitor, with a binding IC50 value of 2.6 nM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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M-808 | 98.72% | M-808 is a highly potent and efficacious covalent Menin-MLL interaction inhibitor, with a binding IC50 value of 2.6 nM. | ||||||||||||||||||||
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