247046-64-6
247046-64-6
Chemical Structure
Dilopetine citrate
Synonym(s): E-6006 citrate
- CAS No.: 247046-64-6
- Formula:C19H27N3O8S
- Molecular Weight:457.50
IUPAC Name: N,N-dimethyl-2-((1-methyl-1H-pyrazol-5-yl)(thiophen-2-yl)methoxy)ethan-1-amine 2-hydroxypropane-1,2,3-tricarboxylate
InChIKey: KRFGVGXHTYATEZ-UHFFFAOYSA-N
SMILES: OC(CC(C(O)=O)(O)CC(O)=O)=O.CN(C)CCOC(C1=CC=CS1)C2=CC=NN2C
Biological Activity: Dilopetine citrate is an inhibitor of substance P release. Dilopetine citrate dose-dependently reduces the vocalizing of isolated guinea pig pups. Dilopetine citrate shows good activity as an antidepressant[1][2].
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Dilopetine citrate | Dilopetine citrate is an inhibitor of substance P release. Dilopetine citrate dose-dependently reduces the vocalizing of isolated guinea pig pups. Dilopetine citrate shows good activity as an antidepressant. | |||||||||||||||||||||
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References
- [1]. Gómez-Gomar A, et al. Enantioseparation of basic pharmaceutical compounds by capillary electrophoresis using sulfated cyclodextrins. Application to E-6006, a novel antidepressant. J Chromatogr A. 2003 Mar 21;990(1-2):91-8. [Content Brief]
- [2]. Hennessy MB, et al. Effects of a novel potential antidepressant on the behavior and cortisol levels of isolated guinea pig pups. Pharmacol Biochem Behav. 2001 Jul-Aug;69(3-4):527-33. [Content Brief]
