2566715-91-9
2566715-91-9
Chemical Structure
KSK68
- CAS No.: 2566715-91-9
- Formula:C23H28N2O2
- Molecular Weight:364.48
InChIKey: XFNQPNJGEZOKCM-UHFFFAOYSA-N
SMILES: O=C(C1CC1)C2=CC=C(OCCCN3CCC(C4=CC=NC=C4)CC3)C=C2
Biological Activity: KSK68 is a high-affinity dual sigma-1 and histamine H3 receptor antagonist, with Kis of 7.7, 3.6, 22.4 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK68 has negligible affinity at the other histamine receptor subtypes. KSK68 can be used for research of nociceptive and neuropathic pain[1].
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KSK68 | KSK68 is a high-affinity dual sigma-1 and histamine H3 receptor antagonist, with Kis of 7.7, 3.6, 22.4 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK68 has negligible affinity at the other histamine receptor subtypes. KSK68 can be used for research of nociceptive and neuropathic pain. | |||||||||||||||||||||
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References
Keywords
