2702280-86-0
2702280-86-0
Chemical Structure
MS117
- CAS No.: 2702280-86-0
- Formula:C17H22N4O
- Molecular Weight:298.38
IUPAC Name: N-(3-(4-(((2-aminoethyl)(methyl)amino)methyl)-1H-pyrrol-3-yl)phenyl)acrylamide
InChIKey: HVDMIAFOVVMNJF-UHFFFAOYSA-N
SMILES: NCCN(C)CC1=CNC=C1C2=CC=CC(NC(C=C)=O)=C2
Biological Activity: MS117 is a first-in-class and cell-active irreversible protein arginine methyltransferase 6 (PRMT6) covalent inhibitor, with an IC50 of 18 nM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
MS117 | 98.0% | MS117 is a first-in-class and cell-active irreversible protein arginine methyltransferase 6 (PRMT6) covalent inhibitor, with an IC50 of 18 nM. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
Keywords
