2702280-86-0
2702280-86-0
Chemical Structure
MS117
- CAS. Nr.: 2702280-86-0
- Formula:C17H22N4O
- Molecular Weight:298.38
IUPAC Name: N-(3-(4-(((2-aminoethyl)(methyl)amino)methyl)-1H-pyrrol-3-yl)phenyl)acrylamide
InChIKey: HVDMIAFOVVMNJF-UHFFFAOYSA-N
SMILES: NCCN(C)CC1=CNC=C1C2=CC=CC(NC(C=C)=O)=C2
Biological Activity: MS117 is a first-in-class and cell-active irreversible protein arginine methyltransferase 6 (PRMT6) covalent inhibitor, with an IC50 of 18 nM[1].
| Art. -Nr. | Produktname | Reinheit | Beschreibung | Pricing | |||||||||||||||||||
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MS117 | 98.0% | MS117 is a first-in-class and cell-active irreversible protein arginine methyltransferase 6 (PRMT6) covalent inhibitor, with an IC50 of 18 nM. | ||||||||||||||||||||
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