2765294-54-8
Chemical Structure
TRPV1 antagonist 3
- CAS No.: 2765294-54-8
- Formula:C23H25N3OS
- Molecular Weight:391.53
IUPAC Name: (S)-N-(3-isopropylphenyl)-2-(5-phenylthiazol-2-yl)pyrrolidine-1-carboxamide
InChIKey: CZISSZWUQQBGMU-FQEVSTJZSA-N
SMILES: CC(C1=CC=CC(NC(N2CCC[C@H]2C3=NC=C(S3)C4=CC=CC=C4)=O)=C1)C
Biological Activity: TRPV1 antagonist 3 (Compound 7q) is a potent TRPV1 antagonist with an IC50 of 2.66 nM against capsaicin. TRPV1 antagonist 3 is mode-selective, oral bioavailable (F = 60%) and CNS-penetrant[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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TRPV1 antagonist 3 | 99.30% | TRPV1 antagonist 3 (Compound 7q) is a potent TRPV1 antagonist with an IC50 of 2.66 nM against capsaicin. TRPV1 antagonist 3 is mode-selective, oral bioavailable (F = 60%) and CNS-penetrant. | ||||||||||||||||||||
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Keywords