3052116-62-5
3052116-62-5
Chemical Structure
CHF-6550
- CAS No.: 3052116-62-5
- Formula:C42H46N4O8
- Molecular Weight:734.84
InChIKey: ZPWHCUCZMYCWNB-WFRZLGIJSA-N
SMILES: O=C(C1=CC=C(C=C1)CNC[C@H](O)C2=C3C=CC(NC3=C(C=C2)O)=O)NCCCOC4=CC=CC([C@](O)(C(O[C@H]5CN(CCC5)C)=O)C6=CC=CC=C6)=C4
Biological Activity: CHF-6550 is an antagonist for muscarinic M3 receptor and an agonist for β2 adrenoceptor (MABA), with pKi of 9.3 and 10.6, respectively. CHF-6550 exhibits good hepatocyte clearance in rat models and good pharmacokinetic characteristics in guinea pigs[1].
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CHF-6550 | CHF-6550 is an antagonist for muscarinic M3 receptor and an agonist for β2 adrenoceptor (MABA), with pKi of 9.3 and 10.6, respectively. CHF-6550 exhibits good hepatocyte clearance in rat models and good pharmacokinetic characteristics in guinea pigs. | |||||||||||||||||||||
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References
Keywords
