473921-12-9
Chemical Structure
Lersivirine
Synonym(s): UK-453061
- CAS No.: 473921-12-9
- Formula:C17H18N4O2
- Molecular Weight:310.35
IUPAC Name: 5-((3,5-diethyl-1-(2-hydroxyethyl)-1H-pyrazol-4-yl)oxy)isophthalonitrile
InChIKey: MCPUZZJBAHRIPO-UHFFFAOYSA-N
SMILES: CCC1=NN(CCO)C(CC)=C1OC2=CC(C#N)=CC(C#N)=C2
Biological Activity: Lersivirine (UK-453061) is potent and selective non-nucleoside reverse transcription inhibitor (NNRTI; IC50=119 nM) with excellent efficacy against NNRTI-resistant viruses. Lersivirine exhibits potent antiretroviral activity against wild-type HIV virus and clinically relevant NNRTI-resistant strains[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Lersivirine | 98.36% | Lersivirine (UK-453061) is potent and selective non-nucleoside reverse transcription inhibitor (NNRTI; IC50=119 nM) with excellent efficacy against NNRTI-resistant viruses. Lersivirine exhibits potent antiretroviral activity against wild-type HIV virus and clinically relevant NNRTI-resistant strains. | ||||||||||||||||||||
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Keywords