MPCI
MPCI is a cell-permeant MC4R-selective ligand with pharmacological chaperone activity. MPCI is a MC4R antagonist with a Ki value of 0.218 μM on HEK293 cells expressing hMC4R. MPCI can be used for the research of MC4R-deficient obesity.
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- CAS No.: 884538-31-2
- Formule: C25H32BrFN4O2
- Masse moléculaire:519.45
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
Description
IC50 & Target
Ki: 0.218 μM (HEK293 cells expressing hMC4R)[1].
Chemical Information
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CAS No. 884538-31-2
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Masse moléculaire 519.45
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Formule C25H32BrFN4O2
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SMILES
O=C(C1=CC=CC(F)=C1CCC2=CC(Br)=CC=C2OC)NC(NCC3CCN(CC3)CC)=N
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)