D2R/D3R/5-HT1AR agonist 1
D2R/D3R/5-HT1AR agonist 1 (compound 22b) is an orally active triple-target D2R/D3R/5-HT1AR agonist with EC50 values of 1.29, 1.05 and 153.5 nM. D2R/D3R/5-HT1AR agonist 1 can improve the behavioral disorders induced by MPTP (HY-W114750) and exerts anti-depression effect. D2R/D3R/5-HT1AR agonist 1 can be used for the research of Parkinson's disease and depression.
For research use only. We do not sell to patients.
- CAS No.: 3028684-07-0
- Formula: C21H35N5O2S
- Molecular Weight:421.60
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
Biological Activity
|
D3 Receptor 1.05 nM (EC50) |
D2 Receptor 1.29 nM (EC50) |
5-HT1A Receptor 153.5 nM (EC50) |
Chemical Information
-
CAS No. 3028684-07-0
-
Molecular Weight 421.60
-
Formula C21H35N5O2S
-
SMILES
O=C(N1CCC(CN([C@@H](CC2)CC3=C2N=C(N)S3)CCC)CC1)N4CCOCC4
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
D2R/D3R/5-HT1AR agonist 1 Related Classifications
HY-179713 Related Classifications
Powered by Bioz