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製品番号: HY-184400

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Pynazolam

Pynazolam is a predicted positive allosteric modulator of GABA_A receptor. 3D-field QSAR and RVM models predict an IC₅₀ of approximately 0.40 nM. Pynazolam can be used in studies related to GABA_A receptor pharmacology.

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CAS 番号: 2034366-97-5
分子式: C₁₆H₁₂N₆O₂
分子量:320.31

保管条件:

Please store the product under the recommended conditions in the Certificate of Analysis.

Pynazolam 構造式

CAS 番号: 2034366-97-5

価格（税別）

Amount: USD 0.00

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

生物活性

製品説明

IC₅₀ & Target

^[1]

GABA_A receptor

体外実験

Pynazolam is predicted to be one of the most active designer benzodiazepines at the GABA-AR, with a log 1/c value of 9.4, indicating potent inhibitory activity in displacing [³H]-diazepam from rat cerebral cortex binding sites^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

化学情報

CAS 番号 2034366-97-5
分子量 320.31
分子式 C₁₆H₁₂N₆O₂
SMILES

O=[N+](C1=CC=C(N2C(CN=C3C4=NC=CC=C4)=NN=C2C)C3=C1)[O-]
輸送条件

Room temperature in continental US; may vary elsewhere.
保管条件

Please store the product under the recommended conditions in the Certificate of Analysis.

純度とドキュメンテーション

取扱説明書 (2659 KB)

参考文献

[1]. Catalani V, et al. In silico studies on recreational drugs: 3D quantitative structure activity relationship prediction of classified and de novo designer benzodiazepines. Chemical biology & drug design. 2023 Jan;101(1):40-51. [Content Brief]

Calculators

モル濃度計算機

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

濃度濃度

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分子量分子量

希釈計算機

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濃度 _(開始) 濃度 _(開始)

体積 _(開始) 体積 _(開始)

濃度 _(終了) 濃度 _(終了)

体積 _(終了) 体積 _(終了)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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MOQ

Minimum order quantity

100 mg

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