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  3. Drug Derivative
  4. PAR4 antagonist 9-phosphoric acid

PAR4 antagonist 9-phosphoric acid is a phosphate prodrug of the PAR4 antagonist 9 (HY-183983). PAR4 antagonist 9-phosphoric acid is applicable to research related to arterial thrombosis.

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PAR4 antagonist 9-phosphoric acid

PAR4 antagonist 9-phosphoric acid Estructura química

No. CAS : 2173066-81-2

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PAR4 antagonist 9-phosphoric acid Related Antibodies

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Descripciòn

PAR4 antagonist 9-phosphoric acid is a phosphate prodrug of the PAR4 antagonist 9 (HY-183983). PAR4 antagonist 9-phosphoric acid is applicable to research related to arterial thrombosis[1].

Parmacokinetics
Species Dose Route AUClast F
Rat[1] 2 mg/kg p.o. 2900 nM·h 21.3 %
In Vivo

PAR4 antagonist 9-phosphoric acid (compound 44) (p.o.) is administered to healthy rats and generates parent compound 32 in vivo, with a relative bioavailability of 44% compared with the optimized formulation of the parent compound[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Peso molecular

672.62

Fòrmula

C29H30FN6O8PS
No. CAS
SMILES

O=C(O[C@@H]([C@@H](OC1=C(F)C=C2N=C(C3=C4N=CC(OCC)=NC4=CC(C)=C3)SC2=C1)C)C)NC5=CN=C(CCOP(O)(O)=O)N=C5
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.
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Referencias
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PAR4 antagonist 9-phosphoric acid Related Classifications

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Keywords:

PAR4 antagonist 9-phosphoric acid2173066-81-2Drug DerivativeDrug derivativeratsfasted-state simulated intestinal fluidhuman liver microsomesphosphate bufferPAR4 receptorplatelet aggregationhuman plateletsγ-thrombinrat liver microsomesarterial thrombosisInhibitorinhibitorinhibit

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Nombre del producto:
PAR4 antagonist 9-phosphoric acid
Cat. No.:
HY-183982
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