PD157672
PD157672 is a selective tachykinin NK3 receptor antagonist. PD157672 can be used for research on central nervous system diseases.
For research use only. We do not sell to patients.
- CAS No.: 159698-59-6
- Formula: C32H47N5O5
- Molecular Weight:581.75
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
[1]|
NK3R |
In Vitro
PD157672, developed via screening and optimization of a dipeptide library, exhibits high selectivity for TACR3[2].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 159698-59-6
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Molecular Weight 581.75
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Formula C32H47N5O5
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SMILES
CC(C)(C)OC(N[C@@H](CC1=CC=CC=C1)C(N[C@](C(NCCCCCCCNC(N)=O)=O)(C)CC2=CC=CC=C2)=O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PD157672 Related Classifications
HY-189102 Related Classifications
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Keywords
- PD157672
- 159698-59-6
- PD 157672
- PD-157672
- Neurokinin Receptor
- smooth muscle contraction
- tachykinin receptor 3
- tachykinin NK2 receptor
- dipeptide library
- guinea pig cortex NK3 receptors
- CNS disorders
- tachykinin NK3 receptor-mediated signaling
- tachykinin NK2 receptor activation
- central and peripheral sites
- TACR3
- Inhibitor
- inhibitor
- inhibit