1. Others GPCR/G Protein Neuronal Signaling
  2. Isotope-Labeled Compounds Adrenergic Receptor
  3. Phentolamine-d4 hydrochloride

Phentolamine-d4 (hydrochloride) is the deuterium labeled Phentolamine hydrochloride. Phentolamine hydrochloride is a reversible, non-selective, and orally active blocker of α1 and α2 adrenergic receptor that expands blood vessels to reduce peripheral vascular resistance. Phentolamine hydrochloride can be used for the research of pheochromocytoma-related hypertension, heart failure and erectile dysfunction[1][2][3].

For research use only. We do not sell to patients.

Phentolamine-d<sub>4</sub> hydrochloride Chemical Structure

Phentolamine-d4 hydrochloride Chemical Structure

CAS No. : 1346599-65-2

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Description

Phentolamine-d4 (hydrochloride) is the deuterium labeled Phentolamine hydrochloride. Phentolamine hydrochloride is a reversible, non-selective, and orally active blocker of α1 and α2 adrenergic receptor that expands blood vessels to reduce peripheral vascular resistance. Phentolamine hydrochloride can be used for the research of pheochromocytoma-related hypertension, heart failure and erectile dysfunction[1][2][3].

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

285.38

Formula

C17H16D4ClN3O

CAS No.
SMILES

N(CC=1NC(C(N1)([2H])[2H])([2H])[2H])(C2=CC(O)=CC=C2)C3=CC=C(C)C=C3.Cl

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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Phentolamine-d4 hydrochloride Related Classifications

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    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Phentolamine-d4 hydrochloride
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HY-12717AS
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