1-(1-[4-[(N-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]piperidin-4- yl)-4H-3,1-benzoxazin-2(1H)-one (L-371,257): a new, orally bioavailable, non-peptide oxytocin antagonist

  • J Med Chem. 1995 Nov 10;38(23):4634-6. doi: 10.1021/jm00023a002.
P D Williams  1 ,  B V Clineschmidt ,  J M Erb ,  R M Freidinger ,  M T Guidotti ,  E V Lis ,  J M Pawluczyk ,  D J Pettibone ,  D R Reiss ,  D F Veber, et al.
Affiliations
  • 1. Department of Medicinal Chemistry, Merck Research Laboratories, West Point, Pennsylvania 19486, USA.
PMID: 7473590 DOI: 10.1021/jm00023a002
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