1 Result for "

EPI7170

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "EPI7170" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-150102
CAS No.: 2139288-26-7
Purity:  99.86%
Target:  

Androgen Receptor

Research Areas:  

Cancer

EPI-7170, a ralaniten analogue, is a potent androgen receptor N-terminal structural domain antagonist that blocks the transcriptional activity of full-length AR (FL-AR) and AR splice variants (AR-Vs). EPI-7170 has antitumor effects against enzalutamide resistant castration-resistant prostate cancer (CRPC) .
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