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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
32 Results for "
N-terminal residue
" in MedChemExpress (MCE) Product Catalog:
Products (32)
32 Results for "N-terminal residue" in MCE Product Catalog:
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27 Publications Verification
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BIX-01294 is a reversible and highly selective G9a and GLP Histone Methyltransferase inhibitor, with IC50s of of 1.7 μM and 0.9 μM, respectively. BIX-01294 inhibits G9a/GLP by competing for binding with the amino acids N-terminal of the substrate lysine residue. BIX-01294, a (1H-1,4-diazepin-1-yl)-quinazolin-4-yl amine derivative, induces necroptosis and autophagy. BIX-01294 has antitumor activity in recurrent tumor cells .
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27 Publications Verification
Cat. No.: HY-108239
CAS No.: 1392399-03-9
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BIX-01294 trihydrochloride is a reversible and highly selective G9a and GLP Histone Methyltransferase inhibitor, with IC50s of of 1.7 μM and 0.9 μM, respectively. BIX-01294 trihydrochloride inhibits G9a/GLP by competing for binding with the amino acids N-terminal of the substrate lysine residue. BIX-01294 trihydrochloride, a (1H-1,4-diazepin-1-yl)-quinazolin-4-yl amine derivative, induces necroptosis and autophagy. BIX-01294 trihydrochloride has antitumor activity in recurrent tumor cells .
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2 Cited Publications
AMP-PCP disodium is an ATP analogue and can bind to Hsp90 N-terminal domain with a Kd value of 3.8 μM. AMP-PCP disodium binding favors the formation of the active homodimer of Hsp90 .
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1 Cited Publications
Synonyms: UDP-N-acetyl-D-galactosamine disodium
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Cat. No.: HY-E70196
CAS No.: 55576-49-3
Synonyms: Asp-N
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Endoproteinase Asp-N (MS grade) is a metalloprotease that can specifically cleave the N-terminal side of aspartyl and cysteic acid residues .
Synonyms: N-Acetyl-L-serine
Cat. No.: HY-P99399
CAS No.: 2159141-27-0
Synonyms: RG 6100; RO7105705; MTAU-9937A
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Cat. No.: HY-P4376A
Cat. No.: HY-P4371
CAS No.: 177942-21-1
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Cat. No.: HY-P1228
CAS No.: 926018-95-3
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Cat. No.: HY-P4371A
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Cat. No.: HY-P1224
CAS No.: 864915-61-7
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Cat. No.: HY-P1230
CAS No.: 852155-81-8
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Cat. No.: HY-P4376
CAS No.: 16869-42-4
Cat. No.: HY-P3692
CAS No.: 1815618-15-5
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Cat. No.: HY-125564
CAS No.: 19245-85-3
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Cat. No.: HY-P1225
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Leucyl aminopeptidase, Porcine is a metallopeptidase that cleave N-terminal residues from proteins and peptides. Leucyl aminopeptidase serves as transcriptional repressors to control pyrimidine, alginate and cholera toxin biosynthesis, as well as mediate site-specific recombination events in plasmids and phages .
Cat. No.: HY-E70691
CLK1 is one of the dual specificity kinases and is the founding member of the 'LAMMER' family of kinases. CLK1 activity is positively regulated by phosphorylation on either tyrosine residues or serine/threonine residues, and is negatively regulated by steric constraints mediated by the N-terminal domain, as well as, by phosphorylation on a subset of serine/threonine residues within the catalytic domain. CLK1 Recombinant Human Active Protein Kinase is a recombinant CLK1 protein that can be used to study CLK1-related functions .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
