3 Results for "

PD134308

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "PD134308" in MCE Product Catalog:

Cat. No.: HY-105226
CAS No.: 130332-27-3
Synonyms: PD134308
Domaines de recherche:  

Neurological Disease Cancer

CI-988 (PD134308) is a potent, selective and orally active CCK2R (cholecystokinin 2 receptor) antagonist with an IC50 of 1.7 nM for mouse cortex CCK2. CI-988 shows >1600-fold selectivity for CCK2 over CCK1 receptor. CI-988 has anxiolytic and anti-tumor effects .
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Cat. No.: HY-105226B
Synonyms: PD134308 hemihydrate
Domaines de recherche:  

Neurological Disease Cancer

CI-988 hemihydrate (PD134308) is a potent, selective and orally active CCK2R (cholecystokinin 2 receptor) antagonist with an IC50 of 1.7 nM for mouse cortex CCK2. CI-988 hemihydrate shows >1600-fold selectivity for CCK2 over CCK1 receptor. CI-988 hemihydrate has anxiolytic and anti-tumor effects .
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Cat. No.: HY-105226A
CAS No.: 130404-91-0
Synonyms: PD134308 meglumin
Domaines de recherche:  

Cardiovascular Disease

CI-988 meglumin is a cholecystokinin 2 receptor (CCK2R) antagonist. CI-988 meglumin prevents the gastrin-mediated protection of the heart with ischemia/reperfusion injury .
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