1 Result for "

UNC9995

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "UNC9995" in MCE Product Catalog:

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1 Cited Publications
Cat. No.: HY-120920
CAS No.: 1354030-52-6
Purity:  99.38%
Target:  

Dopamine Receptor

Research Areas:  

Inflammation/Immunology

UNC9995 is a β-arrestin2-biased agonist of dopamine receptor Drd2. UNC9995 inhibits NLRP3 inflammasome activation by enhancing β-arrestin2-NLRP3 interaction, thus prevents neuronal degeneration. Futhermore, UNC9995 activates the Drd2/β-arrestin2 signaling to prevent inflammation-related genes transcription-induced by JAK/STAT3. UNC9995 improves depressive behavior in mouse model, and improves astrocytes dysfunctions .
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